Cytochrome P450 Drug Interactions Exam Review A+ 2023-2024 1 / 4 1. CYP1A2 Sub- strates 2. CYP1A2 In- hibitors 3. CYP1A2 Induc- ers 4. CYP2C9 Sub- strates 5. CYP2C9 In- hibitors 6. CYP2C9 Induc- ers 7. CYP2C19 Sub- strates 8. CYP2C19 In- hibitors 9. CYP2C19 Induc- ers Amitriptyline (Elavil) Duloxetine (Cymbalta) Ciprofloxacin- Oral (Cipro, Cipro XR) Ciprofloxacin- Otic (Cetraxal, Otiprio) -smoking - St. Johns Wort Carvedilol (Coreg, Coreg CR) Celecoxib (Celebrex) Amiodarone (Cordarone, Pacerone) Fluconazole (Diflucan) Metronidazole (Flagyl) -phenobarbital -phenytoin -St. Johns Wart Citalopram (Celexa) Clopidogrel (Plavix) Esomeprazole (Nexium) Phenytoin (Dilantin) Eslicarbazepine (Zebinix, Aptiom) Esomeprazole (Nexium) Fluconazole (Diflucan) Fluoxetine (Prozac, Sarafem) Fluvoxamine (Luvox) Omeprazole (Prilosec) Ticlopidine (Ticlid) Voriconazole (Vfend, Pfizer) -Carbamazepine (Tegretol) -Phenytoin - Rifampin -St. Johns wortCytochrome P450 Drug Interactions Exam Review A+ 2023-2024 2 / 4 10. CYP2D6 Sub- strates 11. CYP2D6 In- hibitors 12. CYP3A4 Sub- strates Amitriptyline (Elavil) Aripiprazole (Abilify) Codeine (Tylenol with Codeine) Duloxetine (Cymbalta) Tamoxifen (Soltamox) Tramadol (ConZip, Ultram, Qdolo) Bupropion (Aplenzin, Forfivo XL, Wellbutrin SR, Wellbutrin XL) Darifenacin (Enablex) Dronedarone (Multaq) Duloxetine (Cymbalta) Fluoxetine (Prozac, Sarafem) Paroxetine (Paxil, Paxil CR) Sertraline (Zoloft) Terbinafine (Lamisl, Silka Cream) Alprazolam (Xanax) Amiodarone (Cordarone, Pacerone) Amlodipine (Norvasc) Atorvastatin (Lipitor) Carbamazepine (Tegretol) Colchicine (Colcrys, Gloperba, Mitigare) Cyclosporine (Restasis,